Four Days, 3 Symposia, 10 Tracks, and More!
Explore Drug Discovery Chemistry 2027

Focused on the discovery and optimization challenges of small-molecule and macrocyclic drug candidates, the 22nd Annual conference explores the critical "middle space" of drug discovery—from hit identification and lead optimization to emerging modalities, AI-enabled design, and translational strategies. Join a community of discovery scientists and share the innovations shaping the next generation of medicines.

TODAY'S SYNTHETIC MOLECULES FOR TOMORROW'S THERAPEUTICS

APRIL 19
Track IconNext-Generation Induced Proximity Modulators
Track IconRNA-Targeted Small Molecule Drug Discovery
Track IconGenerative AI for Drug Discovery
Track IconView In-Person Training Seminar
Short Courses
APRIL 20 - 21
Track IconDegraders & Molecular
Glues - Part 1
Track IconSmall Molecule Discovery Technologies
Track IconAI/ML for Early Drug Discovery - Part 1
Track IconInnovative Linker & Bioconjugation Chemistries
Track IconOral & Macrocyclic Peptides - Part 1
APRIL 21 - 22
Track IconDegraders & Molecular
Glues - Part 2
Track IconTargeting Protein-Protein Interactions
Track IconAI/ML for Early Drug Discovery - Part 2
Track IconDNA-Encoded Libraries
Track IconOral & Macrocyclic Peptides - Part 2